Tacrolimus CAS 104987-11-3 yog cov tshuaj tiv thaiv kab mob macrolides muaj zog. Ntawm qib molecular, nws cov nyhuv yog kho los ntawm cov protein FKBP12 hauv cytoplasm uas khi nrog nws. FKBP12 ua rau Tacrolimus mus rau hauv lub xovtooj ntawm tes thiab tsim ib qho nyuaj uas sib tw tshwj xeeb rau calmodulin thiab inhibits calmodulin (tom kawg kho calcium-dependent inhibitory signal transduction system nyob rau hauv T-hlwb), thiaj li yuav thaiv tau ib series Gene transcription ntawm lymphokine. Cov kev sim hauv vitro qhia tau hais tias Tacrolimus yog qhov muaj zog tiv thaiv kab mob, nws tuaj yeem cuam tshuam kev tsim ntawm cytotoxic lymphocytes, thiab allograft rejection yog feem ntau tshwm sim los ntawm yav tas los.

Khoom: Tacrolimus CAS 104987-11-3
Lwm Lub Npe: FK506; Kev kawm; Advagraf; Astagraf XL; Envarsus XR; Tacrolimus; CAS 104987-11-3; Tacrolimus API; Advagraf API; Protopic API;
Lub npe tshuaj: (3S, 4R, 5S, 8R, 9E, 12S, 14S, 15R, 16S, 18R, 19R, 26aS)-5, 6, 8, 11, 12, 13, 14, 15, 16, 17, 18, 19, 24, 25, 26, 26a-Hexadecahydro-5, 19-dihydroxy-3-{(1E)-2-[(1R, 3R, 4R){ {37}}hydroxy-3-methoxycyclohexyl]-1-methylethenyl}-14, 16-dimethoxy-4, 10, 12, 18-tetramethyl{46 }}(2-propenyl)-15, 19-epoxy-3H-pyrido[2, 1-c][1, 4]oxaazacyclotricosine{{56} }, 7, 20, 21 (4H, 23H)-tetrone.
Cov mis mos molecular: C44H69TSIS MUAJ12S
Molecular hnyav: 804.02
CAS Nr.: 104987-11-3
Kev ua si lom neeg: Tacrolimus nthuav tawm cov haujlwm lom lom neeg tseem ceeb, feem ntau yog cov tshuaj tiv thaiv kab mob. Nws lub luag haujlwm tseem ceeb ntawm kev ua haujlwm yog inhibition ntawm T-cell activation, uas ua lub luag haujlwm tseem ceeb hauv kev tiv thaiv kab mob.
Cov tshuaj no inhibits kev ua haujlwm ntawm T-hlwb, TH-cell-dependent B-cells-propagation, thiab tiam ntawm lymphokine xws li nthuav qhia ntawm interleukin 2, interleukin 3, -interferon thiab interleukin 2 receptor. Tacrolimus tuaj yeem inhibit allograft rejection ntawm daim tawv nqaij, lub plawv, lub raum thiab daim siab, ncua sij hawm ciaj sia taus ntawm allograft, thiab qhov no yog pov thawj nyob rau hauv lub cev ntawm nas, dev, primate thiab tib neeg. Nws tau dav siv rau kev mob thiab mob ntev ntawm daim siab, lub raum thiab cov pob txha pob txha hloov pauv.
1. Lub sijhawm them nyiaj
TT, LC
2. Hnub xa khoom
Sib tham tau
3. Kev ua lag luam
Middle East / Africa / Asia / South America / Europe
4. Qauv
Muaj
5. Cov qauv kev tswj hwm
CP, EP, USP
6. Daim ntawv pov thawj tsim nyog
Kev tso npe ntawm "A" xwm txheej, Suav GMP; WC daim ntawv tso cai, daim ntawv pov thawj COPP, daim ntawv pov thawj CEP, US DMF tus lej sau npe; MFDS Registration Certificate
7. Ntim me me specification
Pem hauv ntej pob: ib txheej polyethylene hnab thiab txhuas ntawv ci hnab.
Cov pob txheej sab nrauv: Tshuaj kho mob txhuas lub raj mis.
Ntim qhov loj: 500g / lub raj mis.
Peb Qhov Zoo
Peb muaj cov chaw ua haujlwm hauv Dubai thiab Is Nrias teb
peb muaj tus kheej txhim khu kev qha & Kev koom tes ntev & kev paub txog lub Hoobkas
Ntau yam khoom rau xaiv los ntawm Tuam Tshoj thiab Is Nrias teb
Peb tuaj yeem kho raws li koj xav tau
Peb tuaj yeem ua OEM & ODM
Peb tuaj yeem muab N-1 rau API
Tacrolimus CAS 104987-11-3 API FAQ
Q: Tacrolimus yog dab tsi?
Q: Tacrolimus ua haujlwm li cas?
Q: Hom kev hloov pauv hloov pauv li cas Tacrolimus tiv thaiv?
Q: Dab tsi yog qhov kev mob tshwm sim ntawm Tacrolimus?
Q: Puas muaj kev cuam tshuam tshuaj nrog Tacrolimus?
Q: Ua li cas Tacrolimus saib xyuas thaum kho?
Q: Puas siv tau Tacrolimus thaum cev xeeb tub lossis pub niam mis?
Cim npe nrov: tacrolimus cas 104987-11-3, Tuam Tshoj tacrolimus cas 104987-11-3 manufacturers, lwm tus neeg, Hoobkas







